Sylvie DUCKI

2022

titre

Design, synthesis and biological evaluation of conformationnally-restricted analogues of E7010 as inhibitors of tubulin assembly (ITA) and vascular disrupting agents (VDA)

auteur

Vassili Prudhomme, Mélissa Cucca, Lionel Nauton, Elsa Andrieu, Mathilde Fereyrolles, Sylvain Lamoine, Clément Michelin, Khalil Bennis, Aurore Collin, Frédéric de Ceuninck, Iuliana Botez, Christophe Mallet, Sylvie Ducki

article

European Journal of Medicinal Chemistry, 2022, 244, pp.114809. ⟨10.1016/j.ejmech.2022.114809⟩

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Journal articles

DOI

DOI : 10.1016/j.ejmech.2022.114809

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2020

titre

TREK1 channel activation as a new analgesic strategy devoid of opioid adverse effects

auteur

Jérôme Busserolles, Ismail Ben Soussia, Laetitia Pouchol, Nicolas Marie, Mathieu Meleine, Maïly Devilliers, Céline Judon, Julien Schopp, Loïc Clémenceau, Laura Poupon, Eric Chapuy, Serge Richard, Florence Noble, Florian Lesage, Sylvie Ducki, Alain Eschalier, Stéphane Lolignier

article

British Journal of Pharmacology, 2020, 177 (20), pp.4782-4795. ⟨10.1111/bph.15243⟩

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Journal articles

DOI

DOI : 10.1111/bph.15243

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2019

titre

Ethnopharmacological survey of plants used in the traditional treatment of pain conditions in Mali

auteur

Ombeline Danton, Aimé Somboro, Baba Fofana, Drissa Diallo, Lassine Sidibé, Catherine Rubat-Coudert, Fabien Marchand, Alain Eschalier, Sylvie Ducki, Pierre Chalard

article

International Journal of Herbal Medicine, 2019, 17-18, pp.100271. ⟨10.1016/j.hermed.2019.100271⟩

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Journal articles

DOI

DOI : 10.1016/j.hermed.2019.100271

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2018

titre

Analgesic molecules interleaved between layered double hydroxide: Exchange versus in situ reaction and release properties

auteur

Théo Rongere, Arthur Langry, Khalil Bennis, Christine Taviot-Guého, Sylvie Ducki, Fabrice Leroux

article

Journal of Solid State Chemistry, 2018, 268, pp.159 - 167. ⟨10.1016/j.jssc.2018.08.043⟩

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Journal articles

DOI

DOI : 10.1016/j.jssc.2018.08.043

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titre

Optimization of the synthesis of a key intermediate for the preparation of glucocorticoids

auteur

Romain Jouve, Vincent Thery, Sylvie Ducki, Julie Helfenbein, Christophe Thiery, Aurélie Job, Elodie Picard, Christophe Mallet, Isabelle Ripoche, Khalil Bennis

article

Steroids, 2018, 137, pp.14 - 21. ⟨10.1016/j.steroids.2018.06.007⟩

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Journal articles

DOI

DOI : 10.1016/j.steroids.2018.06.007

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2017

titre

Development of the First Two-Pore Domain Potassium Channel TWIK-Related K + Channel 1-Selective Agonist Possessing in Vivo Antinociceptive Activity

auteur

Delphine Vivier, Ismail Ben Soussia, Nuno Rodrigues, Stéphane Lolignier, Maïly Devilliers, Franck Claude Chatelain, Laetitia Prival, Eric Chapuy, Geoffrey Bourdier, Khalil Bennis, Florian Lesage, Alain Eschalier, Jérôme Busserolles, Sylvie Ducki

article

Journal of Medicinal Chemistry, 2017, 60 (3), pp.1076-1088. ⟨10.1021/acs.jmedchem.6b01285⟩

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Journal articles

DOI

DOI : 10.1021/acs.jmedchem.6b01285

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2016

titre

Phthalocyanine-chalcone conjugates

auteur

Fallia Aribi, Charlene Vey, Derya Topkaya, Sinem Tuncel Kostakoglu, Jérémie Fournier-Dit-Chabert, Sebile Işik Büyükekşi, Gökçe Canan Taşkin, Serkan Alpugan, Florian Albrieux, Ayşe Gül Gürek, Mélissa Cucca, Khalil Bennis, Devrim Atilla, Vefa Ahsen, Sylvie Ducki, Fabienne Dumoulin

article

Journal of Porphyrins and Phthalocyanines, 2016, 20, pp.497-504. ⟨10.1142/S1088424616500310⟩

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Journal articles

DOI

DOI : 10.1142/S1088424616500310

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titre

Perspectives on the Two-Pore Domain Potassium Channel TREK-1 (TWIK-Related K+ Channel 1). A Novel Therapeutic Target?

auteur

Delphine Vivier, Khalil Bennis, Florian Lesage, Sylvie Ducki

article

Journal of Medicinal Chemistry, 2016, 59, pp.5149-5157. ⟨10.1021/acs.jmedchem.5b00671⟩

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Journal articles

DOI

DOI : 10.1021/acs.jmedchem.5b00671

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2015

titre

Biochemical investigations of the mechanism of action of small molecules ZL006 and IC87201 as potential inhibitors of the nNOS-PDZ/PSD-95-PDZ interactions.

auteur

Anders Bach, Søren W. Pedersen, Liam A. Dorr, Gary Vallon, Isabelle Ripoche, Sylvie Ducki, Lu-Yun Lian

article

Scientific Reports, 2015, 5, pp.12157. ⟨10.1038/srep12157⟩

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DOI

DOI : 10.1038/srep12157

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2014

titre

Synthesis and structure-activity relationship study of substituted caffeateesters as antinociceptive agents modulating the TREK-1 channel.

auteur

Nuno Rodrigues, Khalil Bennis, Delphine Vivier, Vanessa Pereira, Franck C. Chatelain, Eric Chapuy, Hemantkumar Deokar, Jérôme Busserolles, Florian Lesage, Alain Eschalier, Sylvie Ducki

article

European Journal of Medicinal Chemistry, 2014, 75, pp.391-402

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2013

titre

Assessing the Dual Activity of a Chalcone-Phthalocyanine Conjugate: Design, Synthesis, and Antivascular and Photodynamic Properties

auteur

Sinem Tuncel, Aurélien Trivella, Devrim Atilla, Khalil Bennis, Huguette Savoie, Florian Albrieux, Laetitia Delort, Hermine H. Billard, Virginie Dubois, Vefa Ahsen, Florence F. Caldefie-Chezet, Claire Richard, Ross W. Boyle, Sylvie Ducki, Fabienne Dumoulin

article

Molecular Pharmaceutics, 2013, 10 (10), pp.3706 - 3716. ⟨10.1021/mp400207v⟩

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DOI

DOI : 10.1021/mp400207v

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titre

Structure-Based Design of PDZ Ligands as Inhibitors of 5-HT2A Receptor/PSD-95 PDZ1 Domain Interaction Possessing Anti-hyperalgesic Activity

auteur

Alexandre Vogrig, Liam Dorr, Naoual Bouzidi, Benjamin Boucherle, Anne-Sophie Wattiez, Elisabeth Cassier, Gary Vallon, Isabelle Ripoche, Isabelle Abrunhosa-Thomas, Philippe Marin, Lionel Nauton, Vincent Thery, Christine Courteix, Lu-Yun Lian, Sylvie Ducki

article

ACS Chemical Biology, 2013, 8, pp.2209-2216. ⟨10.1021/cb400308u⟩

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DOI

DOI : 10.1021/cb400308u

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titre

Identification of PDZ ligands by docking-based virtual screening for the development of novel analgesic agents

auteur

Naoual Bouzidi, Hemantkumar Deokar, Alexandre Vogrig, Benjamin Boucherle, Isabelle Ripoche, Isabelle Abrunhosa-Thomas, Liam Dorr, Anne-Sophie Wattiez, Lu-Yun Lian, Philippe Marin, Christine Courteix, Sylvie Ducki

article

Bioorganic and Medicinal Chemistry Letters, 2013, 23, pp.2624-2627. ⟨10.1016/j.bmcl.2013.02.100⟩

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DOI

DOI : 10.1016/j.bmcl.2013.02.100

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2012

titre

Towards dual photodynamic and antiangiogenic agents: design and synthesis of a phthalocyanine-chalcone conjugate.

auteur

Sinem Tuncel, Jérémie Fournier-Dit-Chabert, Florian Albrieux, Vefa Ahsen, Sylvie Ducki, Fabienne Dumoulin

article

Organic & Biomolecular Chemistry, 2012, 10, pp.1154-1157

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2011

titre

NMR evaluation of interactions between substituted-indole and PDZ1 domain of PSD-95

auteur

Alexandre Vogrig, Benjamin Boucherle, I. Ripoche, I. Abrunhosa-Thomas, Lu-Yun Lian, Hemantkumar Deokar, Sylvie Ducki

article

Bioorganic and Medicinal Chemistry Letters, 2011, 21 (11), pp.3349-3353. ⟨10.1016/j.bmcl.2011.04.011⟩

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Journal articles

DOI

DOI : 10.1016/j.bmcl.2011.04.011

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